Synthesis of Analogues of Thyrotropin-Releasing Hormone

The synthesis of ten new thyrotropin-releasing hormone analogues (15-24) which contain uncoded amino acids (L- and D-homoleucine, L- and D-homophenylalanine, L-homoproline and 6-ketopipecolic acid) is described here. The peptide bond formation was achieved in solution phase using pentafluorophenyl e...

Teljes leírás

Elmentve itt :
Bibliográfiai részletek
Szerzők: Somlai Csaba
Baláspiri L
Dokumentumtípus: Cikk
Megjelent: 1994
Sorozat:JOURNAL FUR PRAKTISCHE CHEMIE-CHEMIKER-ZEITUNG 336 No. 6
Tárgyszavak:
doi:10.1002/prac.19943360609

mtmt:1880328
Online Access:http://publicatio.bibl.u-szeged.hu/31990
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520 3 |a The synthesis of ten new thyrotropin-releasing hormone analogues (15-24) which contain uncoded amino acids (L- and D-homoleucine, L- and D-homophenylalanine, L-homoproline and 6-ketopipecolic acid) is described here. The peptide bond formation was achieved in solution phase using pentafluorophenyl ester activation of the N-protected amino acids. The analogues were tested for their ability to release thyrotropin and for CNS activities and proved to be fully inactive. 
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